Anestezol suppositories instructions: composition, form, action, indications, contraindications, recommendations

Anestezol is a drug produced in the form of suppositories intended for rectal use. The product is highly effective and safe. Due to the inclusion of active components in the antihemorrhoidal drug, pain is eliminated, the intensity of bleeding is reduced, inflammation is eliminated, and an anti-inflammatory effect is achieved. The product is produced in a convenient form, which ensures maximum availability of the active component directly to the site of inflammation. The drug has a fast action. The drug does not have a negative effect on liver and kidney function.

pharmachologic effect

Anestezol has local anesthetic, anti-inflammatory and antiseptic effects.

Pharmacodynamics

Anesthesin is able to quickly suppress pain at the local level and relax spasmodic muscles.

The winning effect is achieved thanks to the substances included in the composition, namely:

Thanks to benzocaine, which exhibits its anesthetic properties, pain receptors are blocked . But this effect will manifest itself only at the level of local impact. The surrounding tissues reduce sensitivity, mainly in the area of the exit sections of the anal area. As a result, the patient’s feeling of fear before the act of defecation disappears, which ensures the free passage of feces.
Dermatol prevents the development of the inflammatory process due to its astringent and drying effect. Inflamed tissues are covered with a soft protective film, which leads to the formation of a barrier against pathogenic flora. As a result, there is no generalization of the infection and no transition of the process to deeper parts. In addition, there is an increase in regenerative processes and an increase in the formation of new cell masses.
Menthol, due to its cooling effect, leads to a decrease in the severity of skin itching and inflammatory reaction . As a result, hemorrhoids decrease in size due to selective stimulation in the nerve endings.
Zinc oxide leads to cleansing of mucous membranes against pathogenic microorganisms. Affected surfaces are disinfected, and regenerative processes in cells are enhanced.

Pharmacokinetics

Anestezol acts primarily at the local level.
Absorption into the blood occurs in small quantities, as well as distribution in the body.
Anestezol bypasses metabolic processes through the liver, which ensures relative safety in use.
Parts of the substance that are absorbed into the systemic circulation are excreted through the kidneys. Some components that can be detected in the systemic circulation can penetrate the placental tissue.

How to insert rectal suppositories correctly

The packaging of Anestezol suppositories includes instructions explaining how to insert the suppositories. You can use the following tips:

If you are inserting the candle yourself, sit down first and then insert it carefully and quickly. You can use another method for inserting suppositories: lie on your side, pull your upper leg towards your chest, and then carefully and quickly insert the suppository into the anus. If it doesn't go in, try to push it further. You can ask another person you trust to insert the candle

To do this, you should lie on your side, stretch your knees to your chest, and relax.

While inserting the candle, some people feel a feeling of coldness, but it quickly dissolves inside.

Sometimes patients refuse to use suppositories because they feel awkward about such treatment. But this is the wrong position, since rectal suppositories give effective results and last for a long time.

Indications for use

Anestezol is used to relieve pain and inflammation in:

Uncomplicated internal hemorrhoids.
Internal hemorrhoids, which were joined by a bacterial infection, added bleeding.
In all stages of external hemorrhoidal changes.
Suspicion of internal developing hemorrhoids.
Thrombosis of hemorrhoids.
Fistula tracts in the outlet sections of the intestine.
Chronic fissures in the anus.

For prophylactic purposes, Anestezol can be used during recovery periods after surgery and to prevent the development of an inflammatory reaction.

It should be borne in mind that for hemorrhoids this should be a comprehensive approach.

Method and dosage

According to the standard guidelines, suppositories are administered 1 twice a day. The average course of treatment is 10 days. If necessary, the duration can be increased to consolidate the therapeutic effect.

To increase the effectiveness of drug therapy, a number of requirements must be met:

It is advisable to administer suppositories after defecation to evenly distribute the active components throughout the intestinal mucous membranes,
before using the drug, it is necessary to toilet the anal area using mild soap and warm water,
Suppositories should be stored in the refrigerator door to preserve their hardness and medicinal properties; this approach will also prevent the suppository from softening under the influence of the heat of the hands and will not lead to partial loss of active substances,
the blister cell should be opened carefully so as not to damage the suppository; if you have difficulty removing it, you can use scissors to cut the suppository along the contour and open the halves,
it is permissible to insert the suppository only with the pointed side; when inserted with a blunt end, there is a high probability of additional injury to painful areas,
To facilitate and speed up the insertion process, you should lie on your left side and bend your knees; the pose reduces the distance between the hand and the anal area and relaxes the round muscle of the anus.

Recommended route of drug administration

after inserting the suppository, it is advisable to lie down for 15 minutes or more to avoid premature leakage of the melted drug,
during therapy, you should cut your nails short or use a fingertip; before insertion, the suppository or finger can be lubricated with Vaseline oil,
To enhance the therapeutic effect and in the presence of external hemorrhoids, the use of suppositories can be combined with the application of ointments to the external area of the anus; you can also partially melt the suppository with your fingers and lubricate the painful areas with the resulting composition.

Video with visual instructions and features of inserting rectal suppositories:

Instructions for use

Anestezol suppositories are administered into the rectal area once or twice a day, depending on the severity of the pathological process and the intensity of the pain syndrome.

In order to use Anestezol, it is necessary to carry out preparatory measures, which consist of:

Preliminary bowel movement. If this procedure cannot be carried out, no additional effort should be made. If there is no bleeding, you can give a cleansing enema.
The volume of injected liquid should not exceed half a liter.
Next, you should toilet the anal area and rectum, for this you can use soap. Whenever possible, gloves are used that can protect the patient from germs.
The patient lies on his right side and takes a position with his legs abducted in his stomach. This position helps the rectum straighten, which improves the administration of Anestezol and its further distribution.
After the suppository is inserted, the patient should lie on his stomach for 20-25 minutes.
The optimal period of use is at night, this is necessary for the best effect of Anestezol on the body.

Use during pregnancy and lactation

Pregnant women are advised to use Anestezol with restrictions, only if the expected benefit outweighs the risk.

Despite the local effect of the drug and the potential safety of Anestezol, its use is not recommended due to the possible accumulation of components. Also theoretically, substances are able to pass through the placental barrier, which could cause effects on the fetus.

While using Anestezol, women who are breastfeeding are recommended to use artificial feeding.

Use in children

Anestezol is not indicated for use in children. The need to use Anestezol can be decided by a specialist. The need for use arises in cases where the potential benefit outweighs the risk.

Pharmacodynamics and pharmacokinetics

The use of candles is accompanied by a number of distinctive features:

the therapeutic effect is achieved in a short time,

high bioavailability of active ingredients,

lack of systemic effect on the body,

ease of use of the drug.

Macrogol, which forms the basis of the drug, ensures uniform distribution of the active ingredients over the surface of the rectum and enhances their therapeutic effect.

The complex composition of the suppositories guarantees several types of therapeutic effects:

Anesthesia. The use of suppositories allows you to get rid of severe pain during the treatment of hemorrhoids and anal fissures. Benzocaine is not absorbed by the intestines and does not affect the general functioning of the body.

Astringent action. Provided by combining bismuth subgallate with zinc oxide. Both substances have synergism and enhance each other’s therapeutic effects. Anestezol effectively eliminates the processes of exudation of inflamed intestinal walls during hemorrhoids and reduces bleeding in the presence of anal fissures.

Regeneration. Active substances accelerate the healing of wound surfaces and restoration of intestinal mucous membranes. Regeneration processes are also enhanced against the background of decreased exudation of the intestinal walls.

Side effects

These pathological conditions can develop when starting to use it independently, without prior examination by a specialist. In addition, this may be the development of allergic manifestations to the use of Anestezol.

Among the main manifestations of adverse reactions to use are:

The appearance of irritation in the skin area.
Development of severe irritation.
After administration, itching and burning in the anal area intensifies.
Stool disorders.
Rashes appear on the skin, which are predominantly polymorphic in nature, but most often it is urticaria.
With long-term use of Anestezol, there is a gradual accumulation of substances, which can lead to methemoglobinemia. As a result, there is a gradual disruption of hemoglobin and its ability to transport oxygen.

Methods for quick pain relief for hemorrhoids at home

Hemorrhoids are an insidious chronic disease, during the period of exacerbation it causes a lot of suffering, interferes with normal life and work, every patient dreams of finding suppositories, ointments or painkillers for hemorrhoids that quickly relieve pain and help them return to normal life. Almost everyone wants to be treated at home using effective traditional or folk methods.

Today, medicine has a wide range of treatments for hemorrhoids.

Of course, it is important not just to alleviate the symptoms, but to eliminate the very cause of the disease. To do this, you need to undergo examination and treatment from a proctologist, but there are situations when you can’t get to the doctor yet, and pain and other symptoms need to be relieved as quickly as possible

Where to begin? First of all, it’s worth thinking about why hemorrhoids worsened and where they came from.

Contraindications

Before prescribing Anestezol, it is necessary to consult with a specialist in order to exclude the development of complications or side effects.

Despite the good tolerance of Anestezol suppositories, the following conditions must be excluded:

The presence of hypersensitivity to any component, as well as a history of an allergic reaction to substances similar in composition or medicinal group.
Pathology of the hematopoietic system, hemoglobinopathies. Anestezol is used with restrictions in children.

Release form and composition

Anestezol is available in the form of rectal suppositories in blister or cell-free packages. One package contains 5 suppositories for rectal administration. One cardboard box contains 1 or 2 packages of Anestezol.

The active ingredients in this product are benzocaine, zinc oxide, bismuth subgallate and menthol. One Anestezol rectal suppository contains the following components:

Benzocaine – 100 mg;
Zinc oxide – 20 mg;
Bismuth subgallate – 40 mg;
Menthol – 4 mg.

Analogs

Aurobin is a combined ointment for rectal use that contains an analgesic and anti-inflammatory component. It is used for varicose hemorrhoidal veins and skin pathologies of the anal area. The average price ranges from 250 to 280 rubles .
Relief . The drug containing lidocaine and fluocortolone promotes a combined effect. Can be used both in the acute period of hemorrhoids and in chronic conditions. The average price ranges from 270 to 320 rubles .
Neo-Anuzol . A complex remedy, with incoming drugs that help not only relieve Elena’s inflamed reaction, but also accelerate the healing process. The price averages 60-90 rubles .
Proctosedyl . A drug that has similar indications for use, but due to the heparin it contains, it can cause bleeding. The average price is 200-230 rubles .
Anuzol . A drug with a predominantly herbal component. Leads to a decrease in pain and a decrease in the severity of the inflammatory reaction. Price from 60 to 80 rubles .
Pilex . A herbal preparation that is most effective against varicose veins. Among the main indications for use will be signs of hemorrhoids and varicocele. When taking it, there are no recorded side effects or clinical overdose, but the effectiveness is somewhat lower in relation to medications. Price from 500 rubles .

Neo-Anuzol

Proctosedyl

Anuzol

Pilex

Applications and dosages

The dosage regimen of the drug is determined on an individual basis. Suppositories are recommended to be used rectally, after cleansing or self-emptying the intestines. The drug is used 1-2 times a day, in doses recommended by a specialist.

for adults

The drug can be used by patients of this age category. Suppositories are recommended to be administered in the morning and evening. A single dose is 1 suppository.

for children

The medicinal composition is used by children over the age of 12 years in doses determined for adult patients. Children under 12 years of age do not use the drug due to the lack of clear information about the safety and effectiveness of the application process.

for pregnant women and during lactation

Women during pregnancy, as well as during breastfeeding, can use the composition if there are indications for use. In most cases, the drug is well tolerated and no adverse reactions are observed. To minimize the likelihood of side effects, it is recommended to follow the dosage regimen recommended by your doctor.