Cefecon suppositories for adults. Instructions for use, price, reviews

Allowed during pregnancy

Allowed during breastfeeding

Allowed for children

Has restrictions for older people

Has limitations for liver problems

Has limitations for kidney problems

Colds have a negative impact on overall well-being. They are accompanied by fever, aching joints, and weakness. To eliminate these symptoms, various drugs with antipyretic and analgesic properties are used. It is necessary to approach the treatment of young children with maximum responsibility.

A child may not always swallow a pill or agree to drink syrup. In such cases, pediatricians recommend using Cefekon suppositories for children. This article contains detailed information about the principle of action and features of the use of the drug.

Conditions for dispensing from pharmacies, price of the drug

The medication is available for purchase by patients without presenting a certified prescription form from a doctor.

Tsefekon suppositories for adults

The cost of packaging the medicine differs in different pharmacies and regions. The average price ranges from 110-170 rubles.

Pharmacodynamics and pharmacokinetics

A combined drug belonging to the group of analgesics and antipyretics. Has analgesic properties. Salicylamide and naproxen are non-steroidal anti-inflammatory substances, while caffeine enhances and regulates excitatory processes in the cerebral cortex.

The drug stimulates metabolic processes in various tissues and organs, including the central nervous system and muscle tissue.

Substances are excreted in urine and feces.

Composition, release form

The medication can be found on the shelves of various pharmacies in the form of suppositories for rectal administration. They have a standard size and shape, white or almost white. Suppositories are packaged in plastic cells of 5 pieces.

The cells are placed in a small cardboard box, in which you can find 2 plates of 5 pieces. The product is accompanied by a description detailing all the nuances of use and possible contraindications for therapy.

The drug contains several active ingredients - naproxen, caffeine, salicylamide. They have the main therapeutic effect. As an auxiliary component, the composition contains a suppository base, which ensures the correct consistency during storage at a certain temperature.

Pharmacological properties

Each form of release of the drug has analgesic, analgesic and antipyretic effects. The product directly affects pain centers, blocking them. At the same time, the components of the drug do not negatively affect the mucous membrane of the gastrointestinal tract and its functioning as a whole.

The action of Cefekon does not lead to significant changes in normal body temperature. The drug is excreted through the kidneys and then through the urethra.

Operating principle and effectiveness

Cefekon suppositories for adults are used because of their high effectiveness in eliminating acute symptoms of inflammatory pathologies. The effectiveness of the product is explained by the presence of several active ingredients with different properties.

The drug has an anti-inflammatory and antipyretic effect, helps to quickly relieve the patient of acute pain of various origins when it suddenly appears.

Each substance in the composition has a specific effect:

• Naproxen belongs to the group of non-steroidal anti-inflammatory components, so it has not only analgesic properties. The substance helps eliminate signs of inflammation by blocking the production of components that provoke such disorders. The effect of the medication is especially pronounced in the area of ​​joints, spinal column, and muscles. The ingredient slows down the progression of the disease, which reduces the risk of complications.
• Salicylamide also belongs to the group of non-steroidal anti-inflammatory ingredients, and therefore enhances the effect of naproxen. When using the medicine, the onset of a therapeutic effect is noted within a few minutes.
• Caffeine in the medication stimulates and helps regulate certain processes in the central nervous system, which increases the effectiveness of therapy. As a result, an improvement in the general condition is observed and the occurrence of systemic negative reactions is prevented.
• The drug helps normalize the patient’s sleep, which is often disturbed during prolonged inflammation and the presence of severe pain.

During treatment, there is an elimination of increased irritability, especially in patients with a history of neurological disorders. The effect of the drug occurs quickly, since after administration into the rectum, the components of the composition are absorbed into the systemic bloodstream and distributed throughout the body.

The components of the composition are concentrated in the cartilage tissue of patients, synovial fluid, and muscle fibers. As a result, high efficiency is noted in the fight against pathologies of the musculoskeletal system. Lower concentrations of the ingredients are found in other tissues and body fluids.

The maximum dose of ingredients in the blood is achieved 1 hour after using a single therapeutic dose. After providing a therapeutic effect, the components of the composition are processed in the liver, and breakdown products are evacuated by the kidneys.

In patients with kidney failure or liver pathologies, the process of processing and removing ingredients slows down. This may negatively affect the therapeutic effect.

Interaction with other drugs

If the child is taking any medications, parents are required to inform the attending physician. The fact is that the simultaneous use of different medications can provoke a deterioration of the condition and negatively affect the functioning of internal organs or systems.

It is not recommended to take Cefekon D simultaneously with Nurofen and other medications that contain paracetamol. This combination can cause toxic liver damage.

Severe intoxication of the child's body is the result of combining rectal suppositories with tricyclic antidepressants, Rifampicin or ethanol. Under the influence of the active substance, the suppository significantly enhances the effect of anticoagulants. In this regard, it is necessary to avoid simultaneous use of these medications. Nephrotoxic effects can result from combination with salicylates.

The hypototoxic effect is reduced when taken simultaneously with cimetidine (inhibitors of microsomal oxidation). The effectiveness of medications that have a uricosuric effect is reduced.

Antiepileptic drugs help reduce the concentration of suppository substances in plasma (up to 60%). If the patient is taking or shortly before the onset of ARVI symptoms was undergoing treatment with drugs, it is necessary to tell a specialist about this. He will be able to select the most safe and effective treatment for a cold. Thus, the risk of negative consequences of drug interactions is reduced.

Indications for use

Cefekon suppositories are used in diagnosing various disorders accompanied by pain.

The drug for adults is indicated in the following cases:

• Toothache of varying intensity.
• Headache and migraine. In this case, the drug can be used as an auxiliary method of therapy.
• Pain due to arthrosis in acute and chronic form. The drug somewhat slows the progression of the pathological condition, but is not used as the only method of therapy.
• Arthritis in acute form, in which there is pain in the joint area, as well as swelling and redness.
• Osteochondrosis in acute form, in which there is pain and impaired mobility of the spinal column.
• Radiculitis in the acute stage.
• Neuritis and neuralgia. The drug helps eliminate acute pain that worries patients with this disorder.
• Herpes zoster in the acute stage. With this disorder, patients experience severe pain, so the drug can be used as an auxiliary component of the composition.
• Colds and viral diseases. The medicine is prescribed as an antipyretic when tablet medications are not used for various reasons.
• Muscle pain, discomfort after injury.
• Severe pain during menstruation.

The drug may be included in the course of therapy for other diseases according to individual indications. It is not often used as the only method of therapy.

Price, where to buy

In Russia, the cost of the medicine is about 95 rubles, in Ukraine – 33 UAH.

• Online pharmacies in RussiaRussia
• Online pharmacies in UkraineUkraine

Pharmacy Dialogue

• Tsefekon N (sup. rect. No. 10) Nizhpharm JSC
  121 rub. order

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Pharmacy24

• Tsefekon N N10 candles VAT "Nizhpharm", Nizhny Novgorod, Russian Federation
  85 UAH. order

Contraindications and adverse reactions

Cefekon suppositories for adults are not used if intolerance to any components of the composition is detected.

There are other barriers to therapy:

• Acute gastritis and gastric ulcer. Despite the lack of impact of the components of the composition on the mucous membranes of the digestive tract, when using the drug in the acute period, the condition may worsen.
• Bleeding from the rectum.
• Acute form of hemorrhoids, presence of anal fissures, nodes.
• Diagnosis of angle-closure glaucoma.
• An uncontrolled form of arterial hypertension, in which a hypertensive crisis is often observed.
• Chronic insomnia, developing against the background of a mental or neurological disorder.
• Failure of the liver and kidneys, accompanied by a deterioration in general condition. With such deviations, the effectiveness of the drug decreases and the process of removing the components of the composition worsens.
• The period of pregnancy and breastfeeding.
• Aspirin asthma, which in most cases develops in patients as a result of uncontrolled use of non-steroidal anti-inflammatory drugs.
• Excessive excitability and disturbance of psycho-emotional balance.
• Severe course of pathologies of the cardiovascular system.

The drug is used with caution in the treatment of elderly patients. The medication is also not prescribed for children under 16 years of age.

Despite the rectal use of suppositories and the absence of irritating effects on the tissues of the digestive tract, the drug can provoke complications from internal organs.

Often complications affect the hematopoietic organs, which provokes pronounced negative reactions and aggravation of the general condition. At the same time, during a laboratory test, a decrease in the level of the most important blood cells is detected.

If complications occur, it is important to immediately stop therapy and visit a doctor who will determine the need to prescribe additional medications to normalize the condition.

When using the product as prescribed, an overdose does not develop. But doctors cannot completely eliminate the risk of its development. If negative symptoms worsen, you should immediately consult a doctor.

General information about the drug

The main component of the drug provides mild anti-inflammatory, antipyretic and analgesic effects. The undeniable advantage of the drug is its release form. Since suppositories are introduced directly into the rectum, they act faster and do not have a negative effect on the mucous membrane of the gastrointestinal tract.

It is worth noting that this remedy is prescribed to children from three months. When used correctly, it gently and within a short amount of time eliminates the unpleasant symptoms of acute respiratory infections and is safe for a fragile child’s body.

Side effects are extremely rare. In general, the drug was well tolerated. Since the medicine does not contain a large number of additives, it rarely causes allergic reactions, which is very important for young children.

Cefekon D is a rectal suppository intended specifically for the treatment of children, so manufacturers took care of the comfort of small patients and made small suppositories. Therefore, there are no problems with the introduction.

Drug group, scope of application

Rectal suppositories are part of the pharmacological group of analgesics-antipyretics and are a non-narcotic drug. Manufacturers used paracetamol as the main active ingredient. MNN: Paracetamol.

Application of Cefekon

In the field of pediatrics, it is used to eliminate signs of influenza, ARVI, and normalize the general condition of a child during the development of a viral infection. Prescribed to children under 3 years of age (100 mg). For patients over three years of age, specialists prescribe medication with a dosage higher than 100 mg, taking into account age and weight.

Release forms and average prices for the drug in Russia

The medication is available in the form of white rectal suppositories. To make it as convenient as possible to select the required dosage, you can purchase Cefekon D in pharmacies with different amounts of the main component. The manufacturing company also produces suppositories for adults. Cefekon N differs from the children's drug in composition (more details about the differences between the drugs will be described below). The drug is prescribed to children over 16 years of age.

The price of children's Cefekon depends not only on the dosage, but also on the region of residence:

Prices may change periodically. The availability of the drug and the exact price must be checked directly at the pharmacy in your city.

Composition and pharmacological properties

The antipyretic and analgesic effect is due to paracetamol (50, 100 or 250 mg), which acts as the main active ingredient. The substance, penetrating into the body, blocks cyclooxygenase. Thus, it has an effect on pain and thermoregulatory centers. Also during the production process, solid fat (vitepsol) is used as a form-containing mass.

The drug is characterized by analgesic and antipyretic properties. The anti-inflammatory effect of the suppository is insignificant. This is due to the fact that paracetamol in areas of inflammation is affected by cellular peroxidases. Under the influence of the components of the product, the indicators of water-electrolyte metabolism do not change and the condition of the gastrointestinal mucosa is not disturbed.

Pharmacological features of paracetamol

Paracetamol is characterized by a high level of absorption. After 40-60 minutes, the peak concentration of the substance is recorded. About 15% binds to plasma proteins.

The metabolic process occurs in the liver. Inactive metabolites are formed as a result of the reaction between paracetamol, sulfates and glucuronic acid. The half-life of drug components lasts from two to three hours. Within 24 hours, 85 to 95% of the drug is excreted from the body in the urine. In its original form, approximately 3% of paracetamol is excreted.

How long does it take for suppositories to start working?

Many parents are concerned about the question of how many minutes the drug takes to act. According to pediatricians, if all rules for administering the suppository are followed, the effect will be noticeable within 20-40 minutes.

It is worth noting that the temperature does not normalize abruptly, but gradually, by about half a degree (from 38.5 to 38).

If the temperature rises sharply, the effectiveness of the candles decreases. This is due to the fact that in such situations there is a spasm of the vessels of the rectum. Therefore, the absorption of paracetamol into the blood becomes impossible. Also, the drug may not reduce the temperature if a small dosage is used to treat children over 4 years of age.

Cefekon N: differences and application features

Cefekon N is prescribed for the manifestation of fever, which is the result of infectious and inflammatory diseases. The drug quickly and effectively eliminates toothache, headaches, and is used for neuralgia, injuries or burns.

The main difference between these dosage forms is the composition. The children's drug contains one active ingredient - paracetamol. And adult suppositories are a combined drug and consist of caffeine, naproxen and salicylomide. It is intended for adults and children over 16 years of age.

The mechanism of action and indications for use of both medications are the same. Since Cefekon N contains caffeine and various additives, it can have a negative effect on an unformed child’s body. Therefore, up to 16 years of age, it is better to use the children's form of this drug.

The instructions for use of Cefekon N indicate that suppositories are inserted into the rectum 1-3 times a day, one suppository at a time. The course of treatment is also 3-5 days. It is advisable to consult a specialist before use. He can also select the most appropriate dosage and treatment regimen.

Instructions for use for adults

Tsefekon suppositories for adults are usually used according to the standard scheme, which involves the rectal administration of a suppository in the amount of 1 piece.

Before use, it is necessary to toilet the external genitalia and wash your hands thoroughly. This will prevent infection and the development of complications.

No more than 3 suppositories are allowed to be administered per day at approximately equal time intervals. The official description indicates that the best effect is achieved after a natural bowel movement or a cleansing enema.

Doctors recommend using suppositories after bowel movements. But if it is impossible to defecate or administer an enema, the product is not prohibited from being used. The duration of the therapeutic course is on average 5 days. The duration is adjusted depending on the patient’s condition and the presence of concomitant abnormalities.

For colds and viral diseases

Diagnosis of such a disorder requires the use of medication to reduce body temperature in the acute period and eliminate muscle pain that appears against the background of fever.

The duration of the therapeutic course should not exceed 3 days. It is especially important to follow this rule when using the product at home. The daily dosage for an adult is 2 suppositories. It is recommended to administer them 1 piece in the morning and evening to achieve pronounced results.

If there is no therapeutic effect, you should visit a doctor. It is prohibited to independently extend the course or increase the daily dose.

For diseases of the musculoskeletal system

Cefekon suppositories for adults with damage to the musculoskeletal system are prescribed in courses of 5 days. The daily norm is usually 2 suppositories, but in case of severe pain it is allowed to increase it to 3 suppositories.

In combination with the medicine, other drugs are usually prescribed, the action of which is aimed at eliminating the cause of the disease. If after 5 days the pain does not disappear, it is not allowed to prolong therapy, nor to increase the dose.

For migraines and headaches

The remedy for diagnosing such a disorder is not used so often. It is usually prescribed to patients when, for various reasons, they cannot take tablet medications.

The duration of treatment for such a disorder usually does not exceed 3 days, since use is only necessary during an attack. 1-2 suppositories per day are enough, which are administered rectally according to the standard scheme.

In combination with suppositories, other agents are usually used to increase the effectiveness of therapy. It is allowed to begin use immediately when the first symptoms of migraine appear.

Overdose

Overdose when used in recommended doses is impossible.

If an overdose occurs, side effects may appear and intensify: bronchospasm , tachycardia , heart failure , dizziness , pain and itching in the rectum, increased pressure, dizziness. diarrhea , tremor , hyperthermia , ringing in the ears , arrhythmias , agitation, drowsiness, frequent urination, irritability, seizures, anxiety, confusion, gastrointestinal bleeding, dehydration, headache, delirium , disorientation are also possible . tactile sensitivity.

It is necessary to stop taking the drug and carry out symptomatic therapy, which should be aimed at maintaining heart activity and reducing blood pressure. You may experience discomfort or itching in the rectum. In this case, you should administer an enema with sunflower oil.

Analogs

If the original medicine is not available in pharmacies or it is impossible to prescribe it, a substitute with similar properties is selected. Analogs may have a different composition and are often available in a different dosage form.

The most effective substitutes:

• Ibuprofen is available in tablet form and has strong analgesic and anti-inflammatory properties. Despite the different dosage form, the medication belongs to the group of non-steroidal anti-inflammatory drugs, helps reduce body temperature and is considered very effective. The tablets work due to the presence of ibuprofen as the main active ingredient. The drug is prescribed for fever, arthrosis and arthritis, osteochondrosis, muscle pain of various origins. Treatment usually lasts no more than 5 days, helps eliminate acute symptoms and improve the condition. The cost of the analogue starts from 50 rubles.
• Analdim - rectal suppositories based on algin and diphenhydramine. The drug not only helps to reduce body temperature, but also has pronounced analgesic properties, which makes it possible to alleviate the condition of patients quite quickly. Suppositories are prescribed mainly when diagnosing a febrile state against the background of an infectious and viral disease, but sometimes they are allowed to be used for muscle pain and discomfort of other origins. The daily dosage and duration of use in each case is determined individually depending on the patient's condition. The cost of candles is 60-90 rubles.
• Nimesil is a preparation based on nimesulide, which is available in powder form for the preparation of a solution taken orally. The drug belongs to the group of non-steroidal anti-inflammatory drugs, which allows it to be used for fever of various origins, pain, and pathologies of the musculoskeletal system. The product is considered very effective, despite the presence of another active ingredient in the composition. It helps not only to get rid of pain, but also blocks the production of components that provoke the inflammatory process. Treatment with an analogue usually lasts no longer than 5 days, as when prescribing the original. The price of the product starts from 50 rubles.
• Acetylsalicylic acid in tablet form is considered the simplest and most accessible substitute, which is actively used in the treatment of patients of all ages. The active component of the same name in the tablets helps eliminate pain, reduces body temperature, additionally thins the blood, and reduces the risk of blood clots. The cost of the analogue is 20-50 rubles.

Despite other dosage forms and the presence of other components in the composition, all analogues have similar properties.

Cefekon is a popular anti-inflammatory suppository that is actively used for the treatment of adults in the presence of pain and acute signs of inflammation. Using the medicine according to the schedule and after a doctor’s prescription helps to avoid the development of complications and get results on the first day of treatment.

special instructions

Treatment of young patients requires maximum care and responsibility. In order not to cause harm to the baby, it is necessary to adhere to the recommendations of the attending physician and take into account special instructions that relate to the use of rectal suppositories.

The drug should not be used if the child’s weight does not exceed 5 kg. The risk of side effects from internal systems or organs is much higher in premature babies. This means that treatment should be carried out under the supervision of a specialist.

To avoid toxic liver damage or signs of overdose, drugs should be used for no longer than five days. If after three days the temperature continues to rise, consultation with a qualified specialist is necessary.

Ibuprofen can be used as a drug substitute in cases where it is not effective enough. Replacement of drugs is carried out with the permission or under the supervision of a qualified specialist.

With increased caution, suppositories are prescribed to children who have been diagnosed with liver disorders. If during the course of treatment a deterioration in the condition of the organ occurs, it is necessary to notify the doctor and stop using this drug.

The speed of psychomotor reactions and the state of the central nervous system do not change under the influence of the medication, provided that the dosage was calculated correctly and the patient followed all the specialist’s recommendations. If there is a need to use suppositories for longer than 5 days, it is necessary to monitor liver function. Only a doctor can extend the course of treatment, taking into account the patient’s condition.